Bioactive Small Molecules
Medchemexpress LLC Fmoc-Lys(Tfa)-OH | 76265-69-5 | 99.8% | 464.43 | 100 G
Fmoc-Lys(Tfa)-OH is a lysine derivative. Amino acids and amino acid derivatives have been commercially used as ergogenic supplements, influencing the secretion of anabolic hormones, fuel supply during exercise, mental performance during stress, and preventing exercise-induced muscle damage. They are recognized as beneficial ergogenic dietary substances.
- Influence the secretion of anabolic hormones.
- Supply fuel during exercise.
- Improve mental performance during stressful tasks.
- Prevent exercise-induced muscle damage.
Enzo Life Sciences Ac-IETD-CHO (5mg). CAS: 191338-86-0
Caspase and granzyme inhibitor. Reversible inhibitor of caspase-6, -8 and granzyme B. Also inhibits caspase-10. Alternative name: Caspase 8 inhibitor (aldehyde), Granzyme B inhibitor (aldehyde). Formula: C21H34N4O10. MW: 502.5. Purity: ≥96% (HPLC). Formulation: Lyophilized. Peptide content: 70-90%. Solubility: Soluble in distilled water at 10 mg/mL and in DMSO at 1 mg/mL. Long Term Storage: -20°C. Use/Stability: Use always fresh solutions.
Medchemexpress LLC HY-103200 5mg Medchemexpress, SR59230A (hydrochloride) CAS:1135278-41-9 Purity:>98%
Medchemexpress, HY-103200 5mg SR59230A (hydrochloride) CAS:1135278-41-9 SR59230A hydrochloride is a potent, selective, and blood-brain barrier penetrating β3-adrenergic receptor antagonist with IC50s of 40, 408, and 648 nM for β3, β1, and β2 receptors, respectively. Purity:>98% Medchemexpress has over 10000 novel life-science reagents, reference compounds, APIs and natural compounds for laboratory and scientific use. Other quantity can also be offered.
Medchemexpress LLC Dithiooxamide (rubeanic acid) | 79-40-3 | 99.9% | 120.20 | 50 G
Dithiooxamide (Rubeanic Acid) is a selective chelating agent and a sulfur-containing analog of Oxamide. It forms stable chelates with various metal ions such as lead, iron, cadmium, manganese, and aluminum. These chelates can be separated, enriched, and detected through adsorption on solid adsorbents or electrode surfaces.
- Acts as a selective chelating agent.
- Sulfur-containing analog of oxamide.
- Forms stable chelates with various metal ions.
- Chelates can be separated, enriched, and detected by adsorption.
Bachem Furin Inhibitor II Trifluoroacetate
Furin Inhibitor II Trifluoroacetate, H-D-Arg-D-Arg-D-Arg-D-Arg-D-Arg-D-Arg-NH2, 673202-67-0, C36H75N25O6, Mr 954.16, 1mg. Hexa-D-arginine amide. Hexa-D-arginine amide is a potent furin inhibitor with a Ki of 0.106 μM. It also inhibited the related convertases PACE4 and prohormone convertase-1 (PC1) with Ki values of 0.58 μM and 13 μM, respectively. The stable hexapeptide exhibited protection against anthrax toxemia in vitro and in vivo.
Medchemexpress LLC HY-B1123 50mg , Auranofin CAS:34031-32-8 Purity:>98%
HY-B1123 50mg Auranofin CAS: 34031-32-8 Auranofin (SKF-39162) is a thioredoxin reductase (TrxR) inhibitor with an IC50 of 0.2 μM. Auranofin exhibits antiviral activity against SARS-CoV21, with a CC50 of 4.2 μM for monkey kidney Vero E6 cells. Purity:>98% Medchemexpress has over 10000 novel life-science reagents, reference compounds, APIs and natural compounds for laboratory and scientific use. Other quantity can also be offered.
Cayman Chemical ANTIBODY D13 5mg
An acylhydrazone antifungal; active against C. neoformans in vitro (MIC80 = 0.06 μg/ml); increases survival in mouse models of C. neoformans, C. albicans, or A. fumigatus infection at 20 mg/kg per day, p.o.
Medchemexpress LLC ATI-2341 TFA | 98.1% | 2256.82 (free base) | 5 MG
ATI-2341 is a potent and functionally selective allosteric agonist of C-X-C chemokine receptor type 4 (CXCR4). This compound activates the inhibitory heterotrimeric G protein (Gi) to promote inhibition of cAMP production and induce calcium mobilization.
- Acts as a biased ligand, favoring Gαi activation over Gα13
- Potent and efficacious mobilizer of bone marrow polymorphonuclear neutrophils (PMNs)
- Potent and efficacious mobilizer of hematopoietic stem and progenitor cells (HSPCs)
Cayman Chemical ANTIBODY EML 425 5mg
An inhibitor of p300 and CBP (IC50s = 2.9 and 1.1 µM, respectively); prevents glucose-induced cataract formation in isolated rat lens at 200 µM
Cayman Chemical 4Carboxybutyld4trIphenylp 5mg
An internal standard for the quantification of (4-carboxybutyl)triphenylphosphonium by GC- or LC-MS
![Medchemexpress LLC 2-[1-(4-chloro-phenyl)-cyclopropyl]-7-iodo-5-oxo-4,5-dihydro-pyrazolo[1,5-a]quinazoline-3-carbonitrile | 2226517-75-3 | 98.2% | C20H12ClIN4O | 10MG](https://assets.fishersci.com/TFS-Assets/CCG/product-images/5000261054.png-250.jpg)
Medchemexpress LLC 2-[1-(4-chloro-phenyl)-cyclopropyl]-7-iodo-5-oxo-4,5-dihydro-pyrazolo[1,5-a]quinazoline-3-carbonitrile | 2226517-75-3 | 98.2% | C20H12ClIN4O | 10MG
Dynapyrazole-A is a selective small-molecule inhibitor that targets the ATPase activity of microtubule-stimulated dynamin, used in biochemical and cellular studies to probe dynamin-dependent membrane trafficking and endocytosis processes.
- Selective inhibitor of microtubule-stimulated dynamin ATPase activity.
- High purity 98.2% suitable for research assays.
- Soluble in DMSO (25 mg/mL); available as 10 mM solution in DMSO.
- Stable as powder at -20°C for extended storage; store solutions at -80°C for best stability.
- Suitable for biochemical and cell biology studies involving dynamin-dependent processes.
Medchemexpress LLC HY-N7378 5mg Medchemexpress, N-Hydroxypipecolic acid CAS:115819-92-6 Purity:>98%
Medchemexpress, HY-N7378 5mg N-Hydroxypipecolic acid CAS:115819-92-6 N-Hydroxypipecolic acid (1-Hydroxy-2-piperidinecarboxylic acid), a plant metabolite and a systemic acquired resistance (SAR) regulator, orchestrates SAR establishment in concert with the immune signal salicylic acid. N-Hydroxypipecolic acid accumulates systemically in the plant foliage in response to pathogen attack. N-Hydroxypipecolic acid induces SAR to bacterial and oomycete infection[2][3]. Purity:>98% Medchemexpress has over 10000 novel life-science reagents, reference compounds, APIs and natural compounds for laboratory and scientific use. Other quantity can also be offered.
Medchemexpress LLC Nylidrin hydrochloride | 849-55-8 | 98.7% | 5 MG
Nylidrin hydrochloride, also known as Buphenine hydrochloride, is an orally active β-adrenergic agonist. This compound demonstrates significant biological activity, including antagonism of NR1A/2B NMDA receptors, reduction of NP, HA, and M1 levels, and antiviral efficacy against H1N1 influenza A viruses. It also shows promise in improving hemorrhagic shock and exhibiting anti-allergic effects.
- Orally active β-adrenergic agonist
- Antagonizes NR1A/2B NMDA receptors (IC50 = 0.18 μM in Xenopus oocytes)
- Reduces levels of NP, HA, and M1
- Demonstrates antiviral activity against multiple H1N1 subtype influenza A viruses
- Improves hemorrhagic shock
- Possesses anti-allergic effects
Cayman Chemical ANTIBODY SPI 112 25mg
A cell-impermeable inhibitor of SHP-2 in cell-free assays (IC50 = 1 µM); selectively inhibits SHP-2 over SHP-1 and PTP1B (IC50s = 18.3 and 14.5 µM, respectively)
Cayman Chemical ANTIBODY ML-354 5mg
A PAR4 antagonist (IC50 = 140 nM) that exhibits 71-fold selectivity for PAR4 over PAR1 (IC50 = 10 μM) in isolated human platelets